A Phase 1a/1b Study Investigating the Safety, Tolerability, Pharmacokinetics, Pharmacodynamics, and Preliminary Antitumor Activity of the CDK4 Inhibitor BGB-43395, Alone or as Part of Combination Therapies in Patients With Metastatic HR+/HER2- Breast Cancer and Other Advanced Solid Tumors

2023-506888-34-00 Protocol BGB-43395-101 Human pharmacology (Phase I) - First administration to humans Ongoing, recruiting

Start 22 May 2024 · Status Ongoing, recruiting · 1 EU/EEA countries · 8 sites · Protocol BGB-43395-101

Overview

Sponsor-declared trial summary

Phase Human pharmacology (Phase I) - First administration to humans
Status Ongoing, recruiting
Participants planned 471
Countries 1
Sites 8

Advanced or metastatic solid tumors including hormone receptor positive (HR+), human epidermal growth factor 2 negative (HER2-) breast cancer

Key facts

Sponsor
BeOne Medicines AG
Participant type
Patients
Age range
18-64 years, 65+ years
Gender
Male and Female
Therapeutic area
Diseases [C] - Neoplasms [C04]
Trial duration
22 May 2024 → ongoing
Decision date (initial)
2024-02-26
Transition trial
No
Low-intervention
No
Rare-disease indication
No
Vulnerable population
Yes

Trial design

CTIS Part I — objectives, methods, condition coding

Conditions and MedDRA coding

Advanced or metastatic solid tumors including hormone receptor positive (HR+), human epidermal growth factor 2 negative (HER2-) breast cancer

VersionLevelCodeTermSystem organ class
21.1 PT 10024627 Liposarcoma 100000004864
21.0 PT 10061451 Colorectal cancer 100000004864
20.0 SOC 10029104 Neoplasms benign malignant and unspecified (incl cysts and polyps) 2
20.0 PT 10025031 Lung adenocarcinoma 100000004864
21.0 PT 10061534 Oesophageal squamous cell carcinoma 100000004864
21.1 PT 10017758 Gastric cancer 100000004864
20.0 LLT 10027150 Melanoma malignant 10029104
20.0 PT 10033128 Ovarian cancer 100000004864
21.0 PT 10060121 Squamous cell carcinoma of head and neck 100000004864
23.0 PT 10083234 Hormone receptor positive breast cancer 100000004864
20.0 PT 10015560 Ewing's sarcoma 100000004864
20.0 PT 10001388 Adrenocortical carcinoma 100000004864
28.0 PT 10085481 Hormone receptor positive HER2 negative breast cancer 100000004864
23.0 PT 10065430 HER2 positive breast cancer 100000004864
21.0 PT 10014733 Endometrial cancer 100000004864
20.0 PT 10060862 Prostate cancer 100000004864

Sponsors and contacts

Sponsor organisations, regulatory contacts, third parties

BeOne Medicines AG

Sponsor organisation
BeOne Medicines AG
Address
Aeschengraben 27
City
Basel
Postcode
4051
Country
Switzerland

Scientific contact point

Organisation
BeOne Medicines AG
Contact name
BeOne Medical Officer

Public contact point

Organisation
BeOne Medicines AG
Contact name
BeOne Medical Officer

Locations

1 EU/EEA country · 8 investigational sites

By country

CountryMS statusPlanned subjectsSites
France Ongoing, recruiting 91 8
Rest of world
Brazil, China, United States, Thailand, New Zealand, Moldova, Republic of, Malaysia, Korea, Republic of, Australia
380

Investigational sites

France

8 sites · Ongoing, recruiting
Centre De Lutte Contre Le Cancer Eugene Marquis
Medical oncology, Avenue La Bataille Flandre Dunkerque, Cs 44229, Rennes Cedex
Institut Bergonie
Medical Oncology, 180 R De Saint Genes, 229 Cours De L Argonne, Bordeaux
Centre Oscar Lambret
Medical Oncology, 3 Rue Frederic Combemale, 59000, Lille
Centre Francois Baclesse
Medical Oncology, 3 Avenue Du General Harris, Cs 45026, Caen Cedex 5
Institut Gustave Roussy
DITEP, 114 Rue Edouard Vaillant, 94800, Villejuif
Institut De Cancerologie De L Ouest
Medical oncology, Bd Du Professeur Jacques Monod, 44800, St Herblain
Institut Curie
Medical Oncology, 26 Rue D Ulm, 75005, Paris
Institut Paoli Calmettes
Medical Oncology, 232 Boulevard De Sainte Marguerite, Bp 156, Marseille

Country notifications

Trial-start, recruitment-start, end and early-termination notifications submitted per Member State

Country Trial startTrial end Recruitment startRecruitment end Early termination
France 2024-05-22 2024-05-31

Application history

9 submissions — initial application plus substantial / non-substantial modifications

#TypeCodeSubmittedReference MSConclusionDecision date
1 INITIAL IN 2023-11-01 France Acceptable
2024-02-19
2024-02-26
2 SUBSTANTIAL MODIFICATION SM-1 2024-03-12 France Acceptable with conditions
2024-06-03
2024-06-03
3 SUBSTANTIAL MODIFICATION SM-2 2024-07-15 France Acceptable
2024-09-30
2024-09-30
4 SUBSTANTIAL MODIFICATION SM-3 2024-10-15 France Acceptable
2024-12-02
2024-12-04
5 SUBSTANTIAL MODIFICATION SM-4 2025-01-16 France Acceptable
2025-02-12
2025-02-26
6 SUBSTANTIAL MODIFICATION SM-5 2025-06-06 France Acceptable with conditions
2025-08-14
2025-08-14
7 SUBSTANTIAL MODIFICATION SM-6 2025-12-10 France Acceptable
2025-12-16
2025-12-16
8 NON SUBSTANTIAL MODIFICATION NSM-1 2025-12-19 France Acceptable
2025-12-16
2025-12-19
9 SUBSTANTIAL MODIFICATION SM-7 2026-03-13 France Acceptable
2026-04-30
2026-06-01