[18F]-olaparib PET; Molecular imaging of DNA damage response by [18F]-olaparib PET

2024-511962-34-00 Protocol 19310 Phase I and Phase II (Integrated) - First administration to humans Authorised, recruitment pending

Status Authorised, recruitment pending · 1 EU/EEA countries · 1 sites · Protocol 19310

Overview

Sponsor-declared trial summary

Phase Phase I and Phase II (Integrated) - First administration to humans
Status Authorised, recruitment pending
Participants planned 10
Countries 1
Sites 1

Head and neck squamous cell carcinoma (HNSCC)

• To assess dosimetry, most optimal time point for imaging (Stage I), and safety of [18F]olaparib PET (Stage I + II). • To determine the correlation between tu-mour [18F]-olaparib uptake and tumour PARP-1 expression levels on tumour biopsy (Stage I + II).

Key facts

Sponsor
Universitair Medisch Centrum Groningen
Participant type
Patients
Age range
18-64 years, 65+ years
Gender
Male and Female
Therapeutic area
Diseases [C] - Neoplasms [C04]
Decision date (initial)
2025-04-22
Transition trial
No
Low-intervention
No
Rare-disease indication
No
Vulnerable population
No
Funding sources
UMCG Cancer Research Fund

External identifiers

EU CT number
2024-511962-34-00
ClinicalTrials.gov
NCT06482307

Trial design

CTIS Part I — objectives, methods, condition coding

Main objective

Scope: Pharmacodynamic, Safety

• To assess dosimetry, most optimal time point for imaging (Stage I), and safety of [18F]olaparib PET (Stage I + II).
• To determine the correlation between tu-mour [18F]-olaparib uptake and tumour PARP-1 expression levels on tumour biopsy (Stage I + II).

Secondary objectives 1

  1. • To evaluate changes in tumour [18F]-olaparib uptake, as a read-out of DNA damage, during treatment with platinum-based chemoradio-therapy, and its correlation with changes in PARP protein expression (Stage II).

Conditions and MedDRA coding

Head and neck squamous cell carcinoma (HNSCC)

Eligibility criteria

Principal inclusion / exclusion criteria as submitted by sponsor

Inclusion criteria 9

  1. Patients >18y, with biopsy-proven HPV-negative HNSCC, or patients >40y with HPV-positive HNSCC and high-risk features (i.e. > 10 smoke packs/year AND ≥N2b)
  2. Treatment with chemoradiotherapy using platinum-based chemotherapy is anticipated
  3. Recent archival tumour tissue (<8 weeks prior to inclusion) should be available with sufficient residual material for determination of tumour PARP1 levels
  4. Presence of a tumour lesion ≥10 mm in diameter
  5. ECOG performance status 0-2
  6. Negative pregnancy test in women with childbearing potential
  7. Life expectancy >3 months
  8. Signed written informed consent and able to comply with the protocol
  9. For stage II only: re-biopsy should be deemed feasible by the investigators (as-sessed by head-and-neck surgeon)

Exclusion criteria 2

  1. Recent treatment with PARP inhibitors or other investigational therapies <30 days.
  2. Presence of significant co-morbidities that make participation in the study undesirable according to the treating physician.

Endpoints

Primary and secondary outcome measures (English text)

Primary endpoints 4

  1. • Dose-activity curves for healthy organs
  2. • Tumour: background ratio at different timepoints post-injection
  3. • AEs until 30 days post-injection
  4. • Correlation between standardised uptake value of [18F]-olaparib in tumour lesions, and PARP1 expression levels determined by immunohistochemistry

Secondary endpoints 2

  1. • Absolute and percentage increase in tumour [18F]-olaparib standardised uptake value after one week of chemoradiation compared to baseline tumour [18F]-olaparib standardised uptake value.
  2. • Correlation between standardised uptake value of [18F]-olaparib in tumour lesions, and PARP1 expression levels determined by immunohistochemistry after one week of chemoradiation.

Investigational products

Investigational medicinal products (IMPs), comparators, placebo, auxiliary

Test 1

Olaparib

PRD11647787 · Product

Active substance
Olaparib
Substance synonyms
AZD-2281, AZD2281
Pharmaceutical form
SOLUTION FOR INJECTION
Route of administration
INTRAVENOUS USE
Authorisation status
Not Authorised
ATC code
V09IX — OTHER DIAGNOSTIC RADIOPHARMACEUTICALS FOR TUMOUR DETECTION
MA holder
UNIVERSITY MEDICAL CENTER GRONINGEN
Paediatric formulation
No
Orphan designation
No

Sponsors and contacts

Sponsor organisations, regulatory contacts, third parties

Universitair Medisch Centrum Groningen

Sponsor organisation
Universitair Medisch Centrum Groningen
Address
Hanzeplein 1
City
Groningen
Postcode
9713 GZ
Country
Netherlands

Scientific contact point

Organisation
Universitair Medisch Centrum Groningen
Contact name
M. van Kruchten

Public contact point

Organisation
Universitair Medisch Centrum Groningen
Contact name
M. van Kruchten

Locations

1 EU/EEA country · 1 investigational sites

By country

CountryMS statusPlanned subjectsSites
Netherlands Authorised, recruitment pending 10 1
Rest of world 0

Investigational sites

Netherlands

1 site · Authorised, recruitment pending
Universitair Medisch Centrum Groningen
Medical Oncology, Hanzeplein 1, 9713 GZ, Groningen

Results and documents

Annex IV summary of results, Annex V layperson summary, and all documents registered in CTIS for this trial

Documents 7 files

Public protocol annexes, IB summaries, regulatory submissions and post-authorisation documents registered in CTIS.

TypeTitleVersion
Protocol (for publication) D1_Protocol 2024-511962-34-00 - for publication 3
Protocol (for publication) F3_Radiation_safety_statement_Olaparib_Quadra 1
Recruitment arrangements (for publication) K1_recruitment procedure NL 2024-511962-34-00 4
Subject information and informed consent form (for publication) L1_SIS and ICF 2024-5114962-34-00 3
Summary of Product Characteristics (SmPC) (for publication) E2_SmPC lynparza-epar-product-information_en 1
Synopsis of the protocol (for publication) D1_Protocol synopsis Dutch 2024-511962-34-00 2
Synopsis of the protocol (for publication) D1_Protocol synopsis English 2024-511962-34-00 2

Application history

1 submissions — initial application plus substantial / non-substantial modifications

#TypeCodeSubmittedReference MSConclusionDecision date
1 INITIAL IN 2025-01-21 Netherlands Acceptable
2025-04-22
2025-04-22