A Phase 1a/1b Study to Investigate the Safety, Tolerability, Pharmacokinetics, Pharmacodynamics, and Preliminary Antitumor Activity of BGB-53038, a Pan-KRAS Inhibitor, as Monotherapy or in Combinations in Patients With Advanced or Metastatic Solid Tumors With KRAS Mutations or Amplification

2024-514704-13-00 Protocol BGB-53038-101 Human pharmacology (Phase I) - First administration to humans Ended

End 23 Apr 2026 · Status Ended · 1 EU/EEA countries · 3 sites · Protocol BGB-53038-101

Overview

Sponsor-declared trial summary

Phase Human pharmacology (Phase I) - First administration to humans
Status Ended
Participants planned 194
Countries 1
Sites 3

Advanced or Metastatic Solid Tumors with KRAS Mutations or Amplifications

Key facts

Sponsor
BeOne Medicines AG
Participant type
Patients
Age range
18-64 years, 65+ years
Gender
Male and Female
Therapeutic area
Diseases [C] - Neoplasms [C04]
Trial duration
completed 23 Apr 2026
Decision date (initial)
2025-04-11
Transition trial
No
Low-intervention
No
Rare-disease indication
No
Vulnerable population
Yes

External identifiers

EU CT number
2024-514704-13-00
ClinicalTrials.gov
NCT06585488

Trial design

CTIS Part I — objectives, methods, condition coding

Conditions and MedDRA coding

Advanced or Metastatic Solid Tumors with KRAS Mutations or Amplifications

VersionLevelCodeTermSystem organ class
20.0 LLT 10079440 Non-squamous non-small cell lung cancer 10029104
27.0 LLT 10058546 Esophageal adenocarcinoma metastatic 10029104
21.1 LLT 10051971 Pancreatic adenocarcinoma 10029104
27.0 LLT 10084871 Gastroesophageal junction cancer metastatic 100000004848
21.0 PT 10061451 Colorectal cancer 100000004864
27.0 PT 10063916 Metastatic gastric cancer 100000004864
27.0 PT 10052358 Colorectal cancer metastatic 100000004864

Sponsors and contacts

Sponsor organisations, regulatory contacts, third parties

BeOne Medicines AG

Sponsor organisation
BeOne Medicines AG
Address
Aeschengraben 27
City
Basel
Postcode
4051
Country
Switzerland

Scientific contact point

Organisation
BeOne Medicines AG
Contact name
BeOne Medical Officer

Public contact point

Organisation
BeOne Medicines AG
Contact name
BeOne Medical Officer

Locations

1 EU/EEA country · 3 investigational sites

By country

CountryMS statusPlanned subjectsSites
Spain Ended 30 3
Rest of world
China, Korea, Republic of, New Zealand, Australia, United States
164

Investigational sites

Spain

3 sites · Ended
Hospital Universitario Fundacion Jimenez Diaz
Oncology, Avenida De Los Reyes Catolicos 2, 28040, Madrid
Hospital Universitari Vall D Hebron
Oncology, Passeig De La Vall D'Hebron 119-129, 08035, Barcelona
Hospital Clinico Universitario De Valencia
Oncology, Avenida Blasco Ibanez 17, 46010, Valencia

Application history

5 submissions — initial application plus substantial / non-substantial modifications

#TypeCodeSubmittedReference MSConclusionDecision date
1 INITIAL IN 2025-01-21 Spain Acceptable
2025-03-17
2025-04-11
2 SUBSTANTIAL MODIFICATION SM-1 2025-05-19 Spain Acceptable
2025-07-07
2025-07-08
3 SUBSTANTIAL MODIFICATION SM-2 2025-07-30 Spain Acceptable
2025-09-12
2025-09-15
4 SUBSTANTIAL MODIFICATION SM-3 2025-10-01 Spain Acceptable
2025-10-02
2025-10-02
5 NON SUBSTANTIAL MODIFICATION NSM-1 2026-04-30 Spain Acceptable
2025-10-02
2026-04-30