A study of the PAN-KRAS inhibitor LY4066434 in participants with KRAS mutant solid tumors.

2024-516733-12-00 Protocol J5Q-OX-JRDA Human pharmacology (Phase I) - First administration to humans Ongoing, recruitment ended

Start 13 May 2025 · Status Ongoing, recruitment ended · 5 EU/EEA countries · 18 sites · Protocol J5Q-OX-JRDA

Overview

Sponsor-declared trial summary

Phase Human pharmacology (Phase I) - First administration to humans
Status Ongoing, recruitment ended
Participants planned 750
Countries 5
Sites 18

Pancreatic Ductal Adenocarcinoma, Non-small Cell Lung Cancer, Colorectal Cancer, Advanced Solid Tumor Metastatic Solid Tumor, PanKRAS.

Key facts

Sponsor
Eli Lilly & Co.
Participant type
Patients
Age range
18-64 years, 65+ years
Gender
Male and Female
Therapeutic area
Diseases [C] - Neoplasms [C04]
Trial duration
13 May 2025 → ongoing
Decision date (initial)
2024-11-20
Transition trial
No
Low-intervention
No
Rare-disease indication
No
Vulnerable population
Yes

External identifiers

EU CT number
2024-516733-12-00
WHO UTN
U1111-1309-9988
ClinicalTrials.gov
NCT06607185

Trial design

CTIS Part I — objectives, methods, condition coding

Conditions and MedDRA coding

Pancreatic Ductal Adenocarcinoma, Non-small Cell Lung Cancer, Colorectal Cancer, Advanced Solid Tumor Metastatic Solid Tumor, PanKRAS.

VersionLevelCodeTermSystem organ class
21.1 LLT 10065252 Solid tumor 10029104

Sponsors and contacts

Sponsor organisations, regulatory contacts, third parties

Eli Lilly & Co.

Sponsor organisation
Eli Lilly & Co.
Address
1 Lilly Corporate Center
City
Indianapolis
Postcode
46285-0001
Country
United States

Scientific contact point

Organisation
Eli Lilly & Co.
Contact name
Eli Lilly & Co.

Public contact point

Organisation
Eli Lilly & Co.
Contact name
Eli Lilly & Co.

Locations

5 EU/EEA countries · 18 investigational sites

By country

CountryMS statusPlanned subjectsSites
Belgium Ongoing, recruitment ended 33 3
France Ended 72 2
Germany Ended 100 5
Italy Ended 50 1
Spain Ongoing, recruitment ended 98 7
Rest of world
China, United States, Japan, Taiwan
397

Investigational sites

Belgium

3 sites · Ongoing, recruitment ended
Cliniques Universitaires Saint-Luc
Oncology, Hippokrateslaan 10, Batiment 54, Sint-Lambrechts-Woluwe
Universitair Ziekenhuis Gent
Oncology, Corneel Heymanslaan 10, 9000, Gent
Institut Jules Bordet
Oncology, Mijlenmeersstraat 90, 1070, Anderlecht

France

2 sites · Ended
Centre Leon Berard
Medical Oncology, 28 Rue Laennec, 69008, Lyon
Institut Gustave Roussy
DITEP Drug Development Department, 114 Rue Edouard Vaillant, 94800, Villejuif

Germany

5 sites · Ended
Asklepios Kliniken Hamburg GmbH
Onkologie und Palliativmedizin, Paul-Ehrlich-Strasse 1, Othmarschen, Hamburg
Krankenhaus Nordwest GmbH
Institut für Klinisch-Onkologische Forschung (IKF), Steinbacher Hohl 2-26, Praunheim, Frankfurt Am Main
Universitaetsklinikum Wuerzburg AöR
Interdisziplinäres Studienzentrum (ISZ) mit ECTU, Josef-Schneider-Strasse 6, Grombuehl, Wuerzburg
SLK-Kliniken Heilbronn GmbH
Medizinische Klinik III, Am Gesundbrunnen 20-26, Neckargartach, Heilbronn
Charite Universitaetsmedizin Berlin KöR
Klinik für Hämatologie und Onkologie, ECTU, Hindenburgdamm 30, Lichterfelde, Berlin

Italy

1 site · Ended
Centro Ricerche Cliniche Di Verona S.r.l.
Oncology Unit, Piazzale Ludovico Antonio Scuro 10, 37134, Verona

Spain

7 sites · Ongoing, recruitment ended
Hospital Universitari Vall D Hebron
Medical Oncology, Passeig De La Vall D'Hebron 119-129, 08035, Barcelona
Institut Catala D'oncologia
Medical Oncology, Avinguda De La Gran Via De L'hospitalet 199-203, 08908, L'hospitalet De Llobregat
Hospital Universitario Ramon Y Cajal
Medical Oncology, Carretera Del Colmenar Viejo Km 9 100, Por El Pardo, Madrid
Hospital Universitario 12 De Octubre
Medical Oncology, Avenida De Cordoba Sn, 28041, Madrid
Hospital Universitario Regional De Malaga
Medical Oncology, Avenida De Carlos De Haya S/N, 29010, Malaga
Hospital General Universitario Gregorio Maranon
Medical Oncology, Calle Del Doctor Esquerdo 46, 28009, Madrid
Hospital Del Mar
Medical Oncology, Passeig Maritim De La Barceloneta 25-29, 08003, Barcelona

Country notifications

Trial-start, recruitment-start, end and early-termination notifications submitted per Member State

Country Trial startTrial end Recruitment startRecruitment end Early termination
Belgium 2025-05-13 2025-08-05 2026-02-19
France 2025-12-01
Germany 2025-07-10 2025-08-07 2026-02-19
Italy 2025-08-04 2025-10-20 2026-02-19
Spain 2025-06-12 2025-08-06 2026-02-19

Application history

10 submissions — initial application plus substantial / non-substantial modifications

#TypeCodeSubmittedReference MSConclusionDecision date
1 INITIAL IN 2024-10-10 Belgium Acceptable with conditions
2024-11-20
2024-11-20
2 SUBSTANTIAL MODIFICATION SM-1 2025-01-30 Belgium Acceptable
2025-02-18
2025-02-18
3 SUBSEQUENT ADDITION OF MSC APP-3 2025-03-05 2025-05-08
4 SUBSEQUENT ADDITION OF MSC APP-4 2025-03-20 Acceptable
2025-02-18
2025-06-04
5 SUBSEQUENT ADDITION OF MSC APP-5 2025-04-04 Acceptable
2025-02-18
2025-06-27
6 SUBSEQUENT ADDITION OF MSC APP-6 2025-04-17 Acceptable
2025-02-18
2025-06-27
7 NON SUBSTANTIAL MODIFICATION NSM-1 2025-07-28 Acceptable
2025-02-18
2025-07-28
8 SUBSTANTIAL MODIFICATION SM-2 2025-08-14 Belgium Acceptable
2025-11-07
2025-11-07
9 SUBSTANTIAL MODIFICATION SM-3 2025-12-23 Belgium Acceptable
2026-02-24
2026-02-24
10 SUBSTANTIAL MODIFICATION SM-4 2026-05-04 Acceptable
2026-06-01
2026-06-03