Effect of dapagliflozin on blood magnesium levels in patients with low magnesium due to HNF1beta-associated kidney disease

2024-518855-43-00 Protocol 112930 Therapeutic confirmatory (Phase III) Ended

End 1 May 2025 · Status Ended · 1 EU/EEA countries · 3 sites · Protocol 112930

Overview

Sponsor-declared trial summary

Phase Therapeutic confirmatory (Phase III)
Status Ended
Participants planned 12
Countries 1
Sites 3

Hypomagnesemia due to HNF1beta mutation

To evaluate the effect of SGLT2 inhibition with dapagliflozin 10mg on serum magnesium in diabetic and non-diabetic patients with HNF1beta-associated renal hypomagnesemia

Key facts

Sponsor
Radboud universitair medisch centrum Stichting
Participant type
Patients
Age range
18-64 years, 65+ years
Gender
Male and Female
Therapeutic area
Diseases [C] - Congenital, Hereditary, and Neonatal Diseases and Abnormalities [C16]
Trial duration
completed 1 May 2025
Decision date (initial)
2024-11-22
Transition trial
Yes
Low-intervention
No
Rare-disease indication
Yes
Vulnerable population
No

External identifiers

EU CT number
2024-518855-43-00
EudraCT number
2022-000596-40

Trial design

CTIS Part I — objectives, methods, condition coding

Main objective

Scope: Therapy

To evaluate the effect of SGLT2 inhibition with dapagliflozin 10mg on serum magnesium in diabetic and non-diabetic patients with HNF1beta-associated renal hypomagnesemia

Conditions and MedDRA coding

Hypomagnesemia due to HNF1beta mutation

Eligibility criteria

Principal inclusion / exclusion criteria as submitted by sponsor

Inclusion criteria 4

  1. Genetically proven HNF1beta disease
  2. Renal hypomagnesemia (serum magnesium < 0.70 mmol/l)
  3. Age 18 - 75 years
  4. Informed consent

Exclusion criteria 8

  1. All other types of diabetes mellitus, including type 1 and type 2 diabetes
  2. History of kidney transplantation
  3. Receiving therapy with an SGLT2 inhibitor within 4 weeks prior to enrolment
  4. Previous intolerance for an SGLT2 inhibitor
  5. Pregnancy or lactation
  6. Use of loop diuretics of thiazide diuretics and inability to discontinue these medications before start of the trial
  7. eGFR < 30ml/min/1,73m2
  8. Patient with severe hepatic impairment (Child-Pugh class C)

Endpoints

Primary and secondary outcome measures (English text)

Primary endpoints 1

  1. Change in serum magnesium

Investigational products

Investigational medicinal products (IMPs), comparators, placebo, auxiliary

Test 1

Dapagliflozin

SUB31650 · Substance

Active substance
Dapagliflozin
Pharmaceutical form
FILM-COATED TABLET
Route of administration
ORAL
Max daily dose
10 mg milligram(s)
Max total dose
10 mg milligram(s)
Max treatment duration
4 Week(s)
Authorisation status
Authorised
ATC code
- — -
Marketing authorisation
-
Paediatric formulation
No
Orphan designation
No
Modified vs. Marketing Authorisation
No

Placebo 1

Placebo

SUB21402 · Substance

Active substance
Placebo
Pharmaceutical form
TABLET
Route of administration
ORAL
Max daily dose
10 mg milligram(s)
Max total dose
10 mg milligram(s)
Max treatment duration
4 Week(s)
Authorisation status
Authorised
ATC code
- — -
Marketing authorisation
-
Paediatric formulation
No
Orphan designation
No
Modified vs. Marketing Authorisation
No

Sponsors and contacts

Sponsor organisations, regulatory contacts, third parties

Radboud universitair medisch centrum Stichting

Sponsor organisation
Radboud universitair medisch centrum Stichting
Address
Geert Grooteplein Zuid 10
City
Nijmegen
Postcode
6525 GA
Country
Netherlands

Scientific contact point

Organisation
Radboud universitair medisch centrum Stichting
Contact name
Maartje Verploegen

Public contact point

Organisation
Radboud universitair medisch centrum Stichting
Contact name
Maartje Verploegen

Locations

1 EU/EEA country · 3 investigational sites

By country

CountryMS statusPlanned subjectsSites
Netherlands Ended 12 3
Rest of world 0

Investigational sites

Netherlands

3 sites · Ended
Radboud universitair medisch centrum Stichting
Nephrology, Geert Grooteplein Zuid 10, 6525 GA, Nijmegen
Erasmus Universitair Medisch Centrum Rotterdam (Erasmus MC)
Nephrology, Dr. Molewaterplein 40, 3015 GD, Rotterdam
Amsterdam UMC Stichting
Endocrinology, De Boelelaan 1117, 1081 HV, Amsterdam

Results and documents

Annex IV summary of results, Annex V layperson summary, and all documents registered in CTIS for this trial

Documents 3 files

Public protocol annexes, IB summaries, regulatory submissions and post-authorisation documents registered in CTIS.

TypeTitleVersion
Protocol (for publication) D1_Research_protocol_DAPA-MAG 4
Recruitment arrangements (for publication) K1_blank_document_Recruitment_arrangements 1
Subject information and informed consent form (for publication) L1_Subject_information_informed_consent_form 5

Application history

1 submissions — initial application plus substantial / non-substantial modifications

#TypeCodeSubmittedReference MSConclusionDecision date
1 INITIAL IN 2024-10-16 Netherlands Acceptable
2024-11-22
2024-11-22