A Phase 1 study of LOXO-435 in Locally Advanced or Metastatic Solid Tumors with FGFR3 Gene Alterations

2022-502755-59-00 Protocol LOXO-FG3-22001 Human pharmacology (Phase I) - First administration to humans Ongoing, recruiting

Start 30 Aug 2023 · Status Ongoing, recruiting · 6 EU/EEA countries · 16 sites · Protocol LOXO-FG3-22001

Overview

Sponsor-declared trial summary

Phase Human pharmacology (Phase I) - First administration to humans
Status Ongoing, recruiting
Participants planned 535
Countries 6
Sites 16

Locally Advanced or Metastatic Solid Tumors with FGFR3 Alterations

Key facts

Sponsor
Eli Lilly & Co.
Participant type
Patients
Age range
18-64 years, 65+ years
Gender
Male and Female
Therapeutic area
Diseases [C] - Neoplasms [C04]
Trial duration
30 Aug 2023 → ongoing
Decision date (initial)
2023-06-28
Transition trial
No
Low-intervention
No
Rare-disease indication
No
Vulnerable population
Yes

External identifiers

EU CT number
2022-502755-59-00
WHO UTN
U1111-1286-3894
ClinicalTrials.gov
NCT05614739

Trial design

CTIS Part I — objectives, methods, condition coding

Conditions and MedDRA coding

Locally Advanced or Metastatic Solid Tumors with FGFR3 Alterations

VersionLevelCodeTermSystem organ class
21.1 LLT 10065252 Solid tumor 10029104

Sponsors and contacts

Sponsor organisations, regulatory contacts, third parties

Eli Lilly & Co.

Sponsor organisation
Eli Lilly & Co.
Address
1 Lilly Corporate Center
City
Indianapolis
Postcode
46285-0001
Country
United States

Scientific contact point

Organisation
Eli Lilly & Co.
Contact name
Patient Advocacy

Public contact point

Organisation
Eli Lilly & Co.
Contact name
Patient Advocacy

Locations

6 EU/EEA countries · 16 investigational sites

By country

CountryMS statusPlanned subjectsSites
France Ongoing, recruiting 27 4
Germany Ongoing, recruiting 7 2
Italy Ongoing, recruiting 8 2
Netherlands Ongoing, recruiting 6 1
Norway Ongoing, recruiting 7 2
Spain Ongoing, recruiting 30 5
Rest of world
Australia, Israel, China, Japan, Canada, United States, Korea, Republic of, United Kingdom
450

Investigational sites

France

4 sites · Ongoing, recruiting
Institut Gustave Roussy
Early drug development, 114 Rue Edouard Vaillant, 94800, Villejuif
Institut Bergonie
Medical Oncology, 229 Cours De L Argonne, 33000, Bordeaux
Centre Leon Berard
Medical Oncology, 28 Rue Laennec, 69008, Lyon
Institut Claudius Regaud
Medical Oncology, 1 Avenue Irene Joliot Curie, 31100, Toulouse

Germany

2 sites · Ongoing, recruiting
Universitaetsklinikum Tuebingen
Internal Medicine, Otfried-Mueller-Strasse 10, Nordstadt, Tuebingen
Klinikum rechts der Isar der TU Muenchen AöR
Urology, Ismaninger Strasse 22, Au-Haidhausen, Munich

Italy

2 sites · Ongoing, recruiting
Fondazione Policlinico Universitario Agostino Gemelli IRCCS
UOC Fase 1, Largo Francesco Vito 1, 00168, Rome
Ospedale San Raffaele S.r.l.
Unità di Oncologia Medica, Via Olgettina 60, 20132, Milan

Netherlands

1 site · Ongoing, recruiting
Erasmus Universitair Medisch Centrum Rotterdam (Erasmus MC)
Medical Oncology, Dr. Molewaterplein 40, 3015 GD, Rotterdam

Norway

2 sites · Ongoing, recruiting
Helse Bergen HF
Haukeland University Hospital - Bergen, Jonas Lies Vei 65, 5021, Bergen
Oslo University Hospital HF
Department of oncology, Taarnbygget, Kirkeveien 166, Oslo

Spain

5 sites · Ongoing, recruiting
Hospital Universitario Hm Sanchinarro
Oncology, Calle Ona 10, 28050, Madrid
Hospital Universitario Marques De Valdecilla
Oncology, 5 Planta, Avenida Valdecilla S/n, Santander
Hospital Universitario 12 De Octubre
Oncology, Bloque D, Avenida De Cordoba S/n, Madrid
Catalan Institute Of Oncology
Oncology, Avinguda Gran Via De L'hospitalet 199-203, 08908, L'hospitalet De Llobregat
MD Anderson Cancer Center
Oncology, Calle De Arturo Soria Nº 270, 28033, Madrid

Country notifications

Trial-start, recruitment-start, end and early-termination notifications submitted per Member State

Country Trial startTrial end Recruitment startRecruitment end Early termination
France 2023-10-05 2024-06-26
Germany 2023-08-30 2024-05-06
Italy 2024-05-22 2024-07-24
Netherlands 2024-03-18 2024-07-04
Norway 2023-12-19 2024-03-12
Spain 2023-10-30 2024-02-21

Application history

14 submissions — initial application plus substantial / non-substantial modifications

#TypeCodeSubmittedReference MSConclusionDecision date
1 INITIAL IN 2023-03-03 Norway Acceptable
2023-06-26
2023-06-28
2 NON SUBSTANTIAL MODIFICATION NSM-1 2023-07-07 Norway Acceptable
2023-06-26
2023-07-07
3 NON SUBSTANTIAL MODIFICATION NSM-2 2023-07-07 Acceptable
2023-06-26
2023-07-07
4 NON SUBSTANTIAL MODIFICATION NSM-3 2023-07-10 Acceptable
2023-06-26
2023-07-10
5 NON SUBSTANTIAL MODIFICATION NSM-4 2023-07-10 Acceptable
2023-06-26
2023-07-10
6 NON SUBSTANTIAL MODIFICATION NSM-5 2023-07-11 Acceptable
2023-06-26
2023-07-11
7 NON SUBSTANTIAL MODIFICATION NSM-6 2023-07-21 Acceptable
2023-06-26
2023-07-21
8 NON SUBSTANTIAL MODIFICATION NSM-7 2023-08-10 Acceptable
2023-06-26
2023-08-10
9 SUBSTANTIAL MODIFICATION SM-1 2023-10-20 Norway Acceptable
2024-01-30
2024-01-30
10 SUBSTANTIAL MODIFICATION SM-2 2024-04-19 Norway Acceptable
2024-06-24
2024-06-25
11 SUBSTANTIAL MODIFICATION SM-3 2024-07-09 Norway Acceptable
2024-08-26
2024-08-26
12 SUBSTANTIAL MODIFICATION SM-4 2025-04-25 Norway Acceptable
2025-07-30
2025-07-30
13 SUBSTANTIAL MODIFICATION SM-5 2025-09-24 Norway Acceptable
2025-11-10
2025-11-12
14 SUBSTANTIAL MODIFICATION SM-6 2026-02-09 Norway Acceptable
2026-04-14
2026-04-14