Effect of antifibrotic therapy on regression of myocardial fibrosis after transcatheter aortic valve implantation (TAVI) in aortic stenosis patients with high fibrotic burden

2024-510869-42-00 Therapeutic exploratory (Phase II) Ended

Start 28 Feb 2022 · End 24 Feb 2026 · Status Ended · 1 EU/EEA countries · 15 sites

Overview

Sponsor-declared trial summary

Phase Therapeutic exploratory (Phase II)
Status Ended
Participants planned 150
Countries 1
Sites 15

aortic stenosis patients with high fibrotic burden

The aim of the study is to evaluate the effect of antifibrotic therapy on regression of myocardial fibrosis after TAVI in patients with baseline high fibrotic burden. Therefore, patients will be treated with Spironolactone in addition to standard of care, Spioronolactone + Dihydralazine in addition to standard of care …

Key facts

Sponsor
Universitaetsmedizin Goettingen
Participant type
Patients
Age range
18-64 years, 65+ years
Gender
Male and Female
Therapeutic area
Diseases [C] - Cardiovascular Diseases [C14]
Trial duration
28 Feb 2022 → 24 Feb 2026
Decision date (initial)
2024-07-26
Transition trial
Yes
Low-intervention
No
Rare-disease indication
No
Vulnerable population
No

External identifiers

EU CT number
2024-510869-42-00
EudraCT number
2019-004244-29

Trial design

CTIS Part I — objectives, methods, condition coding

Main objective

Scope: Therapy, Efficacy

The aim of the study is to evaluate the effect of antifibrotic therapy on regression of myocardial fibrosis after TAVI in patients with baseline high fibrotic burden. Therefore, patients will be treated with Spironolactone in addition to standard of care, Spioronolactone + Dihydralazine in addition to standard of care or according to standard of care alone without any study medication. First, differences between patients in the control arm and patients randomized to anti-fibrotic therapy will be analyzed. The second analysis will determine, whether dihydralazine medication in addition to spironolactone is able to increase a potential antifibrotic effect. Myocardial fibrosis will be assessed by cardiac magnetic resonance imaging (CMR) before TAVI and 1 year after. Quantification of potentially irreversible replacement fibrosis will be carried out by late gadolinium enhancement (LGE), and quantification of the potentially reversible diffuse interstitial fibrosis will be performed by measurement of the extracellular volume fraction (ECV), thereby deriving matrix volume and cell volume.

Conditions and MedDRA coding

aortic stenosis patients with high fibrotic burden

VersionLevelCodeTermSystem organ class
20.1 PT 10002906 Aortic stenosis 100000004866

Eligibility criteria

Principal inclusion / exclusion criteria as submitted by sponsor

Inclusion criteria 4

  1. Male, female age ≥ 60
  2. Diagnosis of severe symptomatic aortic stenosis
  3. Transcatheter aortic valve implantation therapy (TAVI) scheduled
  4. Written informed consent

Exclusion criteria 17

  1. Pre-existing dilative or ischemic heart disease with EF<35% and guideline indication for spironolactone
  2. Patient on current medication with spironolactone, eplerenone, or dihydralazine
  3. Presence of coexistent myocardial pathology such as cardiac amyloidosis, hypertrophic cardiomyopathy, or myocarditis
  4. Presence of coexistent severe aortic regurgitation or severe mitral stenosis
  5. Previous surgical valve replacement or repair
  6. Pacemaker or ICD implanted
  7. Renal impairment (serum creatinine > 1,8 mg/dl and/ or GFR < 30 ml/min/1,73 m² BSA)
  8. Significant hypotension (blood pressure < 90 mm Hg systolic and/or < 50 mm Hg diastolic
  9. Serum potassium > 5,1 mmol/l
  10. Contraindications for Spironolactone (anuria, acute renal failure, serum creatinine > 1.8 mg/dl, hyperkalemia, pregnancy)
  11. Contraindications for Dihydralazine (known allergy or hypersensitivity, systemic lupus erythematodes, adrenocortical disorders)
  12. Known active malignant disease with life expectancy < 1 year
  13. Women with child-bearing potential
  14. Simultaneous participation (including a waiting period of 4 weeks) in other interventional clinical trials
  15. Patient without legal capacity who is unable to understand the nature, significance and consequences of the trial
  16. Person who is in a relationship of dependence/employment with the sponsor or the investigator
  17. Known planned operations or catheter-based interventions (e.g. PCI, transcatheter edge-to-edge mitral or tricuspid valve repair) during 3 months after study inclusion; the performance of e.g. PCI immediately before study enrolment and before TAVI is possible

Endpoints

Primary and secondary outcome measures (English text)

Primary endpoints 1

  1. Differences between treatment groups in reduction of extracellular volume (ECV)- derived matrix volume (measured by CMR) after 12 months

Investigational products

Investigational medicinal products (IMPs), comparators, placebo, auxiliary

Test 2

Aldactone® 25, 25 mg überzogene Tabletten

PRD918036 · Product

Active substance
Spironolactone
Pharmaceutical form
COATED TABLET
Route of administration
ORAL
Max daily dose
25 mg milligram(s)
Max total dose
9125 mg milligram(s)
Max treatment duration
12 Month(s)
Authorisation status
Authorised
ATC code
C03DA01 — SPIRONOLACTONE
Marketing authorisation
6618622.00.00
MA holder
ESTEVE PHARMACEUTICALS GMBH
MA country
Germany
Paediatric formulation
No
Orphan designation
No
Modified vs. Marketing Authorisation
No

Nepresol®, 25 mg Tabletten

PRD387556 · Product

Pharmaceutical form
TABLET
Route of administration
ORAL
Max daily dose
50 mg milligram(s)
Max total dose
18250 mg milligram(s)
Max treatment duration
12 Month(s)
Authorisation status
Authorised
ATC code
C02DB01 — DIHYDRALAZINE
Marketing authorisation
5036.00.00
MA holder
TEOFARMA S.R.L.
MA country
Germany
Paediatric formulation
No
Orphan designation
No
Modified vs. Marketing Authorisation
No

Sponsors and contacts

Sponsor organisations, regulatory contacts, third parties

Universitaetsmedizin Goettingen

Sponsor organisation
Universitaetsmedizin Goettingen
Address
Robert-Koch-Strasse 40, Weende Weende
City
Goettingen
Postcode
37075
Country
Germany

Scientific contact point

Organisation
Universitaetsmedizin Goettingen
Contact name
Florian Walker

Public contact point

Organisation
Universitaetsmedizin Goettingen
Contact name
Florian Walker

Locations

1 EU/EEA country · 15 investigational sites

By country

CountryMS statusPlanned subjectsSites
Germany Ended 150 15
Rest of world 0

Investigational sites

Germany

15 sites · Ended
Klinikum der Universitaet Muenchen AöR
Medizinische Klinik und Poliklinik I, Marchioninistrasse 15, Hadern, Munich
Universitaetsklinikum Heidelberg AöR
Klinik für Kardiologie, Angiologie und Pneumologie, Im Neuenheimer Feld 410, Neuenheim, Heidelberg
Vincentius-Diakonissen-Kliniken gAG
Klinik für Kardiologie, Intensivmedizin und Angiologie, Suedendstrasse 32, Suedweststadt, Karlsruhe
Universitaetsklinikum Schleswig-Holstein AöR
Medizinischen Klinik II (Kardiologie, Angiologie und Intensivmedizin), Campus Lübeck, Ratzeburger Allee 160, 23538, Luebeck
Universitaetsklinikum Frankfurt AöR
Medizinischen Klinik III, Kardiologie, Theodor-Stern-Kai 7, 60590, Frankfurt Am Main
University Medical Center Hamburg-Eppendorf
Universitäteres Herz- und Gefäßzentrum Hamburg, Klinik für Kardiologie, Martinistrasse 52, Eppendorf, Hamburg
Herzzentrum Leipzig GmbH
Universitätsklinik für Kardiologie, Struempellstrasse 39, Probstheida, Leipzig
Universitaetsmedizin Goettingen
Kardiologie und Pneumolog, Robert-Koch-Strasse 40, Weende, Goettingen
Charite Universitaetsmedizin Berlin KöR
Klinik für Kardiologie, Angiologie und Intensivmedizin, Campus Virchow-Klinikum, Augustenburger Platz 1, Wedding, Berlin
Deutsches Herzzentrum Muenchen Des Freistaates Bayern Klinik An Der Technischen Universitaet Muenchen
Klinik für Herz- und Kreislauferkrankungen, Lazarettstrasse 36, Neuhausen-Nymphenburg, Munich
Charite Universitaetsmedizin Berlin KöR
Experiamental and Clinical Research Center (ECRC) Kardiologie Campus Buch, Lindenberger Weg 80, Buch, Berlin
Universitaetsmedizin der Johannes Gutenberg-Universitaet Mainz KöR
Zentrum für Kardiologie, Langenbeckstrasse 1, Oberstadt, Mainz
Kerckhoff-Klinik GmbH
Klinik für Kardiologie und Pneumlogie, Benekestrasse 2-8, 61231, Bad Nauheim
Technical University Of Munich School Of Medicine
Medizinische Klinik und Poliklinik Innere Medizin I - Kardiologie, Ismaninger Strasse 22, Au-Haidhausen, Munich
Charite Universitaetsmedizin Berlin KöR
Medizinische Klinik für Kardiologie CBF, Hindenburgdamm 30, Lichterfelde, Berlin

Country notifications

Trial-start, recruitment-start, end and early-termination notifications submitted per Member State

Country Trial startTrial end Recruitment startRecruitment end Early termination
Germany 2022-02-28 2026-02-24 2022-03-21 2024-07-24

Results and documents

Annex IV summary of results, Annex V layperson summary, and all documents registered in CTIS for this trial

Documents 6 files

Public protocol annexes, IB summaries, regulatory submissions and post-authorisation documents registered in CTIS.

TypeTitleVersion
Protocol (for publication) D1_Reduce-MFA_CTP_for pub 9
Recruitment arrangements (for publication) Reduce-MFA_Document not applicable acc to Clinical Trials Directive EC No 200120EC 1
Subject information and informed consent form (for publication) L1_Reduce-MFA_PatInfo_for Pub 4.2
Subject information and informed consent form (for publication) L1_Reduce-MFA_PIC_Biomaterialsammlung_for Pub 1
Summary of Product Characteristics (SmPC) (for publication) G_FI_Aldactone_25_Spironolacton_Feb_2022 2.0
Summary of Product Characteristics (SmPC) (for publication) G_FI_Nepresol_25_Dihydralazin _ Juni_2015 1

Application history

3 submissions — initial application plus substantial / non-substantial modifications

#TypeCodeSubmittedReference MSConclusionDecision date
1 INITIAL IN 2024-07-09 Germany Acceptable
2024-07-19
2024-07-26
2 SUBSTANTIAL MODIFICATION SM-1 2024-09-16 Germany Acceptable
2024-11-07
2024-11-07
3 NON SUBSTANTIAL MODIFICATION NSM-1 2025-06-27 Germany Acceptable
2024-11-07
2025-06-27