A Phase 1a/b Study Investigating the Safety, Tolerability, Pharmacokinetics, Pharmacodynamics, and Preliminary Antitumor Activity of PRMT5 Inhibitor BGB-58067 Alone and in Combination with Anticancer Agents in Patients With Advanced Solid Tumors

2024-515307-19-00 Human pharmacology (Phase I) - First administration to humans Ongoing, recruiting

Start 24 Mar 2025 · Status Ongoing, recruiting · 3 EU/EEA countries · 10 sites

Overview

Sponsor-declared trial summary

Phase Human pharmacology (Phase I) - First administration to humans
Status Ongoing, recruiting
Participants planned 580
Countries 3
Sites 10

Advanced, or metastatic solid tumors with methylthioadenosine phosphorylase (MTAP) homozygous deletion and/or lost MTAP protein expression

Key facts

Sponsor
BeOne Medicines AG
Participant type
Patients
Age range
18-64 years, 65+ years
Gender
Male and Female
Therapeutic area
Diseases [C] - Neoplasms [C04]
Trial duration
24 Mar 2025 → ongoing
Decision date (initial)
2025-07-18
Transition trial
No
Low-intervention
No
Rare-disease indication
No
Vulnerable population
Yes

External identifiers

EU CT number
2024-515307-19-00
ClinicalTrials.gov
NCT06589596

Trial design

CTIS Part I — objectives, methods, condition coding

Conditions and MedDRA coding

Advanced, or metastatic solid tumors with methylthioadenosine phosphorylase (MTAP) homozygous deletion and/or lost MTAP protein expression

VersionLevelCodeTermSystem organ class
20.0 LLT 10028982 Neoplasm biliary tract 10029104
20.0 PT 10018338 Glioma 100000004864
20.0 LLT 10079440 Non-squamous non-small cell lung cancer 10029104
21.1 LLT 10025734 Malignant neoplasm of biliary tract part unspecified 10029104
21.0 LLT 10033600 Pancreatic adenocarcinoma non-resectable 10029104
24.0 LLT 10085300 Squamous non-small cell lung cancer 100000004848
21.0 LLT 10049280 Solid tumour 10029104
28.0 PT 10089216 PD-L1 protein expression 100000004848
21.1 PT 10061873 Non-small cell lung cancer 100000004864
27.0 PT 10059515 Non-small cell lung cancer metastatic 100000004864
27.0 PT 10008593 Cholangiocarcinoma 100000004864
20.0 PT 10073364 Ductal adenocarcinoma of pancreas 100000004864
27.0 PT 10063157 Metastatic glioma 100000004864

Sponsors and contacts

Sponsor organisations, regulatory contacts, third parties

BeOne Medicines AG

Sponsor organisation
BeOne Medicines AG
Address
Aeschengraben 27
City
Basel
Postcode
4051
Country
Switzerland

Scientific contact point

Organisation
BeOne Medicines AG
Contact name
BeOne Medical Officer

Public contact point

Organisation
BeOne Medicines AG
Contact name
BeOne Medical Officer

Locations

3 EU/EEA countries · 10 investigational sites

By country

CountryMS statusPlanned subjectsSites
Denmark Ongoing, recruiting 9 1
France Ongoing, recruiting 40 5
Spain Ongoing, recruiting 30 4
Rest of world
Korea, Republic of, Australia, United States, China
501

Investigational sites

Denmark

1 site · Ongoing, recruiting
Rigshospitalet
Oncology, Blegdamsvej 9, 2100, Copenhagen Oe

France

5 sites · Ongoing, recruiting
Institut Bergonie
Medical oncology, 180 R De Saint Genes, 229 Cours De L Argonne, Bordeaux
Institut Curie
Department of Drug Development and Innovation (D3i), 26 Rue D Ulm, 75005, Paris
Institut Gustave Roussy
Department of Drug Development, 114 Rue Edouard Vaillant, 94800, Villejuif
Institut De Cancerologie De L Ouest
Medical Oncology, Boulevard Jacques Monod, 44805, Saint-Herblain Cedex
Institut Paoli Calmettes
oncology department, 232 Boulevard De Sainte Marguerite, Bp 156, Marseille

Spain

4 sites · Ongoing, recruiting
Hospital Clinico San Carlos
Oncology, Calle Del Profesor Martín Lagos S/n, 28040, Madrid
Hospital Universitario Hm Sanchinarro
Oncology, Calle Ona 10, 28050, Madrid
Hospital Universitario Fundacion Jimenez Diaz
Oncology, Avenida De Los Reyes Catolicos 2, 28040, Madrid
Hospital Universitari Vall D Hebron
Oncology, Passeig De La Vall D'Hebron 119-129, 08035, Barcelona

Country notifications

Trial-start, recruitment-start, end and early-termination notifications submitted per Member State

Country Trial startTrial end Recruitment startRecruitment end Early termination
Denmark 2025-08-06 2025-08-06
France 2025-07-09 2025-07-09
Spain 2025-03-24 2025-03-24

Application history

8 submissions — initial application plus substantial / non-substantial modifications

#TypeCodeSubmittedReference MSConclusionDecision date
1 INITIAL IN 2024-10-25 France Acceptable
2025-01-24
2025-01-29
2 SUBSTANTIAL MODIFICATION SM-1 2025-02-18 France Acceptable 2025-04-16
3 SUBSEQUENT ADDITION OF MSC APP-3 2025-03-14 2025-05-22
4 SUBSTANTIAL MODIFICATION SM-2 2025-04-17 France Acceptable 2025-05-19
5 SUBSTANTIAL MODIFICATION SM-3 2025-06-30 France Acceptable
2025-07-15
2025-07-15
6 SUBSTANTIAL MODIFICATION SM-5 2025-08-04 France Acceptable
2025-09-26
2025-09-26
7 SUBSTANTIAL MODIFICATION SM-6 2025-12-15 France Acceptable
2026-03-25
2026-03-31
8 NON SUBSTANTIAL MODIFICATION NSM-1 2026-04-20 France Acceptable
2026-03-25
2026-04-20