A study to test how well different doses of BI 1815368 are tolerated by healthy men

2023-503815-13-00 Protocol 1485-0002 Human pharmacology (Phase I) - Other Ended

Start 19 Jun 2023 · End 6 Jun 2024 · Status Ended · 1 EU/EEA countries · 1 sites · Protocol 1485-0002

Overview

Sponsor-declared trial summary

Phase Human pharmacology (Phase I) - Other
Status Ended
Participants planned 60
Countries 1
Sites 1

Healthy

Key facts

Sponsor
Boehringer Ingelheim International GmbH
Participant type
Healthy volunteers
Age range
18-64 years
Gender
Male
Therapeutic area
Diseases [C] - Eye Diseases [C11]
Trial duration
19 Jun 2023 → 6 Jun 2024
Decision date (initial)
2023-05-30
Transition trial
No
Low-intervention
No
Rare-disease indication
No
Vulnerable population
No

Trial design

CTIS Part I — objectives, methods, condition coding

Conditions and MedDRA coding

Healthy

VersionLevelCodeTermSystem organ class
21.0 LLT 10053349 Pharmacokinetic study 10022891

Sponsors and contacts

Sponsor organisations, regulatory contacts, third parties

Boehringer Ingelheim International GmbH

Sponsor organisation
Boehringer Ingelheim International GmbH
Address
Binger Strasse 173
City
Ingelheim Am Rhein
Postcode
55216
Country
Germany

Scientific contact point

Organisation
Boehringer Ingelheim International GmbH
Contact name
CT Disclosure & Data Transparency

Public contact point

Organisation
Boehringer Ingelheim International GmbH
Contact name
CT Disclosure & Data Transparency

Locations

1 EU/EEA country · 1 investigational sites

By country

CountryMS statusPlanned subjectsSites
Belgium Ended 60 1
Rest of world 0

Investigational sites

Belgium

1 site · Ended
SGS Belgium
Clinical Pharmacology Unit Antwerpen, Drie Eikenstraat 655, 2650, Edegem

Country notifications

Trial-start, recruitment-start, end and early-termination notifications submitted per Member State

Country Trial startTrial end Recruitment startRecruitment end Early termination
Belgium 2023-06-19 2024-06-06 2023-06-23 2024-04-30

Oversight and notifications

Regulatory notifications under CTR Articles 38, 52, 53, 54 and 77

Temporary halts 1 · Art. 38 CTR

Temporary halt TH-4196

Halt date
2023-08-18
Member states concerned
Belgium
Publication date
2023-08-25
Reason
Safety related (clinical or pre-clinical results)
Explanation
In the second dose group (150 mg BID) all 8 subjects receiving BI 1815368 have showed increased serum creatinine (up to a max of 1.44 mg/dl (normal range 0.67 – 1.17 mg/dl) and decrease estimated glomerular filtration rate (GFR) (based on creatinine). Other routine labs were normal. The sponsor instructed the site to stop further dosing to all subjects in the trial until the relevance of the above-mentioned findings can be fully evaluated, and appropriate monitoring can be established.
Follow-up measures
All subjects have been tested for additional parameters to evaluate renal function which include cystatin c, urea and urinalyses.
As of 21st of August all subjects remained asymptomatic and levels of creatinine are improving after drug discontinuation. Additional investigations of renal function (urea and urinalysis) remained within normal limits. Results of Cystatin-C are still pending.
Benefit-risk balance changed
No
Treatment stopped
Yes

Application history

3 submissions — initial application plus substantial / non-substantial modifications

#TypeCodeSubmittedReference MSConclusionDecision date
1 INITIAL IN 2023-04-05 Belgium Acceptable
2023-05-30
2023-05-30
2 SUBSTANTIAL MODIFICATION SM-1 2023-10-11 Belgium Acceptable
2023-11-14
2023-11-16
3 SUBSTANTIAL MODIFICATION SM-2 2024-03-05 Belgium Acceptable
2024-04-12
2024-04-15